SCHEMBL8008712

SCHEMBL8008712

CCCCCCCCC=CCCCCCCCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.62
CDC25A P30304 10/20 0.57
CES1 P23141 2/20 0.57
FAAH O00519 2/20 0.56
ALDH1A1 P00352 1/20 0.55
ALDH2 P05091 1/20 0.55
ALDH3A1 P30838 1/20 0.55
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008707 1.00 MGLL (0.62) MGLLCDC25ACES1FAAHALDH1A1
SCHEMBL12664538 0.97 MGLL (0.61) MGLLCDC25ACES1FAAHALDH1A1
SCHEMBL30958386 0.97 MGLL (0.61) MGLLCDC25ACES1FAAHALDH1A1
SCHEMBL28985362 0.95 MGLL (0.55) MGLLCDC25ACES1FAAHALDH1A1
SCHEMBL23731163 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL8863074 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL10725536 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL732925 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL6050334 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL8863090 0.90 CES1 (0.68) CDC25ACES1ALDH1A1ALDH2ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958658-A MECHANICALLY FORMING DROPLETS OF AN ETHYLENICALLY UNSATURATED MONOMER AND A HYDROPHOBIC GROUP HAVING LOG P(CALC) GREATER THAN LOG P(CALC) OF UNSATURATED MONOMER BY ATLEAST ONE UNIT AND WATER INSOLUBLE LUBRICANT, POLYMERIZING, COTAING, DRYING EASTMAN KODAK COMPANY (US) 1999-09-28 US claimed
US-5866312-A MULTILAYER; SUPPORT, SILVER HALIDE EMULSION LAYER AND LIGHT INSENSITIVE OVERCOATING OF HYDROPHILIC BINDER AND POLYMER PARTICLES EASTMAN KODAK COMPANY (US) 1999-02-02 US claimed
US-5858634-A MECHANICALLY FORMING VERY SMALL DROPLETS OF UNSATURATED MONOMER; POLYMERIZING; COATING WITH BINDER; DRYING EASTMAN KODAK COMPANY (US) 1999-01-12 US claimed
EP-0886178-A1 Photographic element having surface protective layer EASTMAN KODAK COMPANY (US) 1998-12-23 EP claimed
EP-0886177-A1 Photographic element containing polymeric particles made by a microsuspension process EASTMAN KODAK COMPANY (US) 1998-12-23 EP claimed
US-6165702-A Imaging element containing polymer particles and lubricant EASTMAN KODAK COMPANY (US) 2000-12-26 US disclosed
EP-0709399-B1 The process for making photographic polymeric matte bead particles EASTMAN KODAK CO (US) 2000-04-05 EP disclosed
US-5981156-A Thermally processable imaging element EASTMAN KODAK COMPANY (US) 1999-11-09 US disclosed
US-5958658-A MECHANICALLY FORMING DROPLETS OF AN ETHYLENICALLY UNSATURATED MONOMER AND A HYDROPHOBIC GROUP HAVING LOG P(CALC) GREATER THAN LOG P(CALC) OF UNSATURATED MONOMER BY ATLEAST ONE UNIT AND WATER INSOLUBLE LUBRICANT, POLYMERIZING, COTAING, DRYING EASTMAN KODAK COMPANY (US) 1999-09-28 US disclosed
US-5866312-A MULTILAYER; SUPPORT, SILVER HALIDE EMULSION LAYER AND LIGHT INSENSITIVE OVERCOATING OF HYDROPHILIC BINDER AND POLYMER PARTICLES EASTMAN KODAK COMPANY (US) 1999-02-02 US disclosed
US-5858634-A MECHANICALLY FORMING VERY SMALL DROPLETS OF UNSATURATED MONOMER; POLYMERIZING; COATING WITH BINDER; DRYING EASTMAN KODAK COMPANY (US) 1999-01-12 US disclosed
EP-0886177-A1 Photographic element containing polymeric particles made by a microsuspension process EASTMAN KODAK COMPANY (US) 1998-12-23 EP disclosed
US-5750328-A POLYMERIC CORE SURROUNDED BY A LAYER OF COLLOIDAL INORGANIC PARTICLES EASTMAN KODAK COMPANY (US) 1998-05-12 US disclosed
EP-0709400-B1 Method of making polymeric particles EASTMAN KODAK CO (US) 1997-12-29 EP disclosed
US-5563226-A FORMING SUSPENSION OF ETHYLENICALLY UNSATURATED MONOMER DROPLETS IN AQUEOUS MEDIA, ADDING GELATIN, AND POLYMERIZING MONOMER EASTMAN KODAK COMPANY (US) 1996-10-08 US disclosed
EP-0709400-A2 Method of making polymeric particles EASTMAN KODAK COMPANY (US) 1996-05-01 EP disclosed
EP-0709399-A2 The process for making photographic polymeric matte bead particles EASTMAN KODAK COMPANY (US) 1996-05-01 EP disclosed
US-5492960-A ADDITION POLYMERIZATION OF ETHYLENICALLY UNSATURATED MONOMER DROPLETS IN AQUEOUS MIXTURE CONTAINING NONREACTIVE COMPOUND AND SURFACTANT OR HYDROPHILIC COLLOID EASTMAN KODAK COMPANY (US) 1996-02-20 US disclosed
US-5455320-A Limited coalescing polymerization of an unsaturated compound and nonreactive compound suspended in water containing a stabilizer EASTMAN KODAK COMPANY (US) 1995-10-03 US disclosed
EP-0653442-A2 Method of making polymeric particles EASTMAN KODAK COMPANY (US) 1995-05-17 EP disclosed