SCHEMBL8008974

SCHEMBL8008974

Cc1ccc(C(C)(C)C)nc1Br

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
TSHR P16473 1/20 0.32
CCR4 P51679 2/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12051879 0.83 TDP1 (0.34) TDP1
SCHEMBL22211759 0.80 HSP90AA1 (0.35) TDP1KDM4E
SCHEMBL12570324 0.78 NOS3 (0.48) NOS3NOS1NOS2TSHRCCR4
SCHEMBL10236287 0.77 NOS3 (0.43) TDP1NOS3NOS1NOS2TSHR
SCHEMBL22624090 0.77
SCHEMBL19143739 0.77 TDP1 (0.33) TDP1
SCHEMBL27756269 0.76 NPC1 (0.32)
SCHEMBL1511034 0.76 ALDH1A1 (0.35) TDP1TSHRKDM4E
SCHEMBL2476935 0.74 NOS3 (0.34) NOS3NOS1NOS2TSHRCCR4
SCHEMBL24917151 0.74 RAB9A (0.34) TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140163-A1 OXAZOLOBENZIMIDAZOLE DERIVATIVES MERCK & CO., INC. (US) 2009-11-19 WO disclosed