SCHEMBL8009717

SCHEMBL8009717

NCC(Cn1ncc2ccc(Sc3ccccc3)cc21)OC(=O)/C=C/C(=O)OC(CN)Cn1ncc2ccc(Sc3ccccc3)cc21

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMO O15229 9/20 0.40
HTR2A P28223 5/20 0.36
HTR2C P28335 5/20 0.36
HTR2B P41595 4/20 0.36
HTR1A P08908 2/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
HTR1D P28221 1/20 0.36
HTR7 P34969 1/20 0.36
HTR4 Q13639 1/20 0.36
ABL1 P00519 1/20 0.32
CXCL12 P48061 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
SIRT3 Q9NTG7 1/20 0.31
EGLN2 Q96KS0 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006857 0.88 HTR2A (0.41) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8007690 0.78 HTR2A (0.40) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL906040 0.75 HTR2A (0.60) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL8007092 0.71 HTR2C (0.48) KMOHTR2AHTR2CHTR2BHTR1A
Ammonia Solution, Strong SCHEMBL906042 0.67 KMO (0.42) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL7777106 0.67 SLC22A12 (0.37) HTR2AHTR2C
Fumaric Acid SCHEMBL8009278 0.67 HTR2A (0.58) KMOHTR2AHTR2CHTR2BHTR1A
Fumaric Acid SCHEMBL8009273 0.67 HTR2A (0.58) KMOHTR2AHTR2CHTR2BHTR1A
Fumaric Acid SCHEMBL8006854 0.67 HTR2A (0.58) KMOHTR2AHTR2CHTR2BHTR1A
SCHEMBL906041 0.64 SLC6A4 (0.36) KMOHTR2AHTR2CHTR2BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000017170-A2 N1-SUBSTITUTED BENZOPYRAZOLES AS INHIBITORS OF 5-HT2 RECEPTORS VERNALIS RESEARCH LIMITED (GB) 2000-03-30 WO disclosed