SCHEMBL8007690

SCHEMBL8007690

CS(=O)(=O)c1ccc2cnn(CC(CN)OC(=O)/C=C/C(=O)OC(CN)Cn3ncc4ccc(S(C)(=O)=O)cc43)c2c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.40
HTR2C P28335 6/20 0.40
HTR2B P41595 4/20 0.40
HTR1A P08908 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
HTR1D P28221 1/20 0.40
HTR7 P34969 1/20 0.40
HTR4 Q13639 1/20 0.40
KMO O15229 7/20 0.39
NAMPT P43490 1/20 0.33
PTGS2 P35354 1/20 0.33
AKR1C3 P42330 2/20 0.32
AKR1C2 P52895 2/20 0.32
CHRM1 P11229 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006857 0.83 HTR2A (0.41) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL8009717 0.78 KMO (0.40) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8009708 0.78 HTR2A (0.56) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8007684 0.78 HTR2A (0.56) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8009714 0.78 HTR2A (0.56) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL8009710 0.74 KMO (0.36) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL8007796 0.70 CA2 (0.42) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL23904366 0.67 NAMPT (0.44) KMONAMPTPTGS2AKR1C3AKR1C2
SCHEMBL7777139 0.63 SLC22A12 (0.39) HTR2AHTR2CHTR2BKMO
SCHEMBL7778328 0.63 ADORA2A (0.34) KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000017170-A2 N1-SUBSTITUTED BENZOPYRAZOLES AS INHIBITORS OF 5-HT2 RECEPTORS VERNALIS RESEARCH LIMITED (GB) 2000-03-30 WO disclosed