SCHEMBL8009818

SCHEMBL8009818

[c]1ccc(Cc2cnc[nH]2)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.67
HRH4 Q9H3N8 4/20 0.67
TAAR1 Q96RJ0 2/20 0.67
CYP3A4 P08684 1/20 0.65
MAPT P10636 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
CYP2D6 P10635 1/20 0.46
ADRA1D P25100 2/20 0.46
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4321538 0.83 HRH3 (0.68) HRH3HRH4TAAR1SMN1; SMN2
Immethridine SCHEMBL29462340 0.80 HRH3 (1.00) HRH3HRH4TAAR1CYP3A4MAPT
Immethridine SCHEMBL30053193 0.78 CYP3A4 (1.00) HRH3HRH4TAAR1CYP3A4MAPT
SCHEMBL28759658 0.77 HRH3 (1.00) HRH3HRH4TAAR1CYP3A4MAPT
SCHEMBL7924408 0.77 HRH3 (1.00) HRH3HRH4TAAR1CYP3A4MAPT
SCHEMBL9783259 0.68 HRH3 (0.73) HRH3HRH4TAAR1CYP3A4MAPT
SCHEMBL320687 0.68 CALM1 (0.44) CYP3A4SMN1; SMN2
SCHEMBL9203875 0.68 MAOA (0.37) HRH3TAAR1
SCHEMBL2626810 0.68 HRH3 (0.65) HRH3HRH4TAAR1CYP3A4MAPT
SCHEMBL10217408 0.68 HRH3 (0.69) HRH3HRH4TAAR1CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US claimed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO claimed
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed