SCHEMBL8009953

SCHEMBL8009953

COc1cc(NC(=O)c2cc(OCCCN(C)C)nn2Cc2ccccc2)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.47
NPSR1 Q6W5P4 3/20 0.46
GAA P10253 1/20 0.44
ACHE P22303 2/20 0.43
BACE1 P56817 1/20 0.43
PDE7A Q13946 1/20 0.42
ATM Q13315 1/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
GUCY1B2 O75343 1/20 0.42
CYP1A2 P05177 1/20 0.42
CHRM2 P08172 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
CYP2D6 P10635 1/20 0.42
CHRM1 P11229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL972626 0.87 NPSR1 (0.52) SMN1; SMN2NPSR1GAAATMMAPT
Hydrochloric Acid SCHEMBL2035215 0.86 NPSR1 (0.51) SMN1; SMN2NPSR1GAAATMMAPT
SCHEMBL8008245 0.86 NPSR1 (0.48) NPSR1GAAMAPTKDM4EGUCY1B2
SCHEMBL8009956 0.85 GRN (0.43) SMN1; SMN2NPSR1GAAACHEMAPT
SCHEMBL8010517 0.84 NPSR1 (0.52) NPSR1GAAMAPTKDM4EGUCY1B2
SCHEMBL8009905 0.84 MAPT (0.54) SMN1; SMN2NPSR1GAAMAPTKDM4E
3,4,5-Trimethoxybenzamide SCHEMBL8009946 0.83 GRN (0.42) SMN1; SMN2NPSR1GAAACHEKDM4E
SCHEMBL7999011 0.83 MET (0.51) NPSR1MAPT
SCHEMBL8013247 0.83 BRD4 (0.51) SMN1; SMN2NPSR1GAAMAPTKDM4E
SCHEMBL8007265 0.82 KDM4E (0.50) SMN1; SMN2MAPTKDM4EGUCY1B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000027394-A1 ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE UNIVERSITY COLLEGE LONDON (GB) 2000-05-18 WO disclosed