SCHEMBL972626

SCHEMBL972626

COc1ccc(NC(=O)c2cc(OCCCN(C)C)nn2Cc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.52
AKR1C3 P42330 2/20 0.46
MAPT P10636 3/20 0.46
KCNJ6 P48051 2/20 0.45
KCNJ3 P48549 2/20 0.45
KCNJ5 P48544 1/20 0.45
LTA4H P09960 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
FAAH O00519 1/20 0.44
ALDH1A1 P00352 2/20 0.44
ATM Q13315 1/20 0.44
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPK1 P28482 1/20 0.43
GAA P10253 1/20 0.43
RECQL P46063 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2035215 0.99 NPSR1 (0.51) NPSR1AKR1C3MAPTKCNJ6KCNJ3
SCHEMBL8010517 0.90 NPSR1 (0.52) NPSR1MAPTKCNJ6KCNJ3LTA4H
SCHEMBL8009940 0.89 ALDH1A1 (0.57) NPSR1MAPTLTA4HMEN1KMT2A
SCHEMBL8009953 0.87 SMN1; SMN2 (0.47) NPSR1MAPTALDH1A1ATMSMN1; SMN2
SCHEMBL8008245 0.86 NPSR1 (0.48) NPSR1MAPTFAAHALDH1A1MAPK1
SCHEMBL8009905 0.85 MAPT (0.54) NPSR1MAPTKCNJ6KCNJ3KCNJ5
SCHEMBL7999011 0.84 MET (0.51) NPSR1MAPTKCNJ6KCNJ3KCNJ5
SCHEMBL8013247 0.84 BRD4 (0.51) NPSR1MAPTFAAHALDH1A1SMN1; SMN2
SCHEMBL8007265 0.83 KDM4E (0.50) MAPTFAAHALDH1A1SMN1; SMN2KDM4E
SCHEMBL7998139 0.83 TRPV1 (0.47) NPSR1MAPTALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 253 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240103007-A1 MASS SPECTROMETRY SAMPLE PROCESSING METHODS, CHROMATOGRAPHY DEVICES, AND DATA ANALYSIS TECHNIQUES FOR BIOMARKER ANALYSIS PROTEAS BIOANALYTICS, INC. (US) 2024-03-28 US claimed
EP-4264274-A1 MASS SPECTROMETRY SAMPLE PROCESSING METHODS, CHROMATOGRAPHY DEVICES, AND DATA ANALYSIS TECHNIQUES FOR BIOMARKER ANALYSIS Proteas Bioanalytics, Inc. (US) 2023-10-25 EP claimed
US-20230087609-A1 USE OF A SOLUBLE GUANYLATE CYCLASE (sGC) STIMULATOR OR OF A COMBINATION OF A sGC STIMULATOR AND AN sGC ACTIVATOR FOR CONDITIONS WHEREIN THE HEME GROUP OF sGC IS OXIDIZED OR WHEREIN sGC IS DEFICIENT IN HEME UNIVERSITEIT MAASTRICHT (NL) 2023-03-23 US claimed
US-20230083417-A1 THERAPEUTIC COMBINATION FOR THE TREATMENT OF BRAIN ISCHEMIA AND SAID THERAPEUTIC COMBINATION FOR USE IN THE TREATMENT OF BRAIN ISCHEMIA UNIVERSITEIT MAASTRICHT (NL) 2023-03-16 US claimed
EP-4110396-A1 THERAPEUTIC COMBINATION FOR THE TREATMENT OF BRAIN ISCHEMIA AND SAID THERAPEUTIC COMBINATION FOR USE IN THE TREATMENT OF BRAIN ISCHEMIA Universiteit Maastricht (NL) 2023-01-04 EP claimed
EP-4106741-A1 USE OF A SOLUBLE GUANYLATE CYCLASE (SGC) STIMULATOR OR OF A COMBINATION OF A SGC STIMULATOR AND AN SGC ACTIVATOR FOR CONDITIONS WHEREIN THE HEME GROUP OF SGC IS OXIDIZED OR WHEREIN SGC IS DEFICIENT IN HEME Universiteit Maastricht (NL) 2022-12-28 EP claimed
US-20220211702-A1 METHODS AND MATERIALS FOR GENDER-DEPENDENT TREATMENT OF CARDIOVASCULAR DYSFUNCTION MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2022-07-07 US claimed
WO-2022132834-A1 MASS SPECTROMETRY SAMPLE PROCESSING METHODS, CHROMATOGRAPHY DEVICES, AND DATA ANALYSIS TECHNIQUES FOR BIOMARKER ANALYSIS PROTEAS BIOANALYTICS, INC. (US) 2022-06-23 WO claimed
CN-114144229-A Methods and materials for gender-dependent treatment of cardiovascular dysfunction 梅约医学教育与研究基金会 2022-03-04 CN claimed
EP-3952992-A1 METHODS AND MATERIALS FOR GENDER-DEPENDENT TREATMENT OF CARDIOVASCULAR DYSFUNCTION Mayo Foundation for Medical Education and Research (US) 2022-02-16 EP claimed
US-20050181066-A1 Novel use of guanylate cyclase activators for the treatment of respiratory insufficiency ALTANA PHARMA AG (DE) 2005-08-18 US claimed
EP-1501605-A1 NOVEL USE OF GUANYLATE CYCLASE ACTIVATORS FOR THE TREATMENT OF RESPIRATORY INSUFFICIENCY ALTANA Pharma AG (DE) 2005-02-02 EP claimed
WO-2003090870-A1 NOVEL USE OF GUANYLATE CYCLASE ACTIVATORS FOR THE TREATMENT OF RESPIRATORY INSUFFICIENCY ALTANA PHARMA AG (DE) 2003-11-06 WO claimed
US-20260116886-A1 DEUTERATED sGC STIMULATORS TISENTO THERAPEUTICS INC (US) 2026-04-30 US disclosed
EP-3532063-B1 COMBINATION THERAPY FOR TREATING PULMONARY HYPERTENSION PULMOKINE INC (US) 2026-03-04 EP disclosed
US-20260000653-A1 TREATMENT OF CNS DISEASES WITH sGC STIMULATORS TISENTO THERAPEUTICS INC (US) 2026-01-01 US disclosed
WO-2008124505-A2 SOLUBLE GUANYLATE CYCLASE (SGC) MODULATORS FOR TREATMENT OF LIPID RELATED DISORDERS IRONWOOD PHARMACEUTICALS,INC. (US) 2008-10-16 WO disclosed
US-20050181066-A1 Novel use of guanylate cyclase activators for the treatment of respiratory insufficiency ALTANA PHARMA AG (DE) 2005-08-18 US disclosed
EP-1501605-A1 NOVEL USE OF GUANYLATE CYCLASE ACTIVATORS FOR THE TREATMENT OF RESPIRATORY INSUFFICIENCY ALTANA Pharma AG (DE) 2005-02-02 EP disclosed
WO-2003090870-A1 NOVEL USE OF GUANYLATE CYCLASE ACTIVATORS FOR THE TREATMENT OF RESPIRATORY INSUFFICIENCY ALTANA PHARMA AG (DE) 2003-11-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260116886-A1 DEUTERATED sGC STIMULATORS PDE2A, PRKG1, GUCY1A2 NPSR1 1857/4885AKR1C3 4422/4885MAPT 4558/4885
US-20230087609-A1 USE OF A SOLUBLE GUANYLATE CYCLASE (sGC) STIMULATOR OR OF A COMBINATION OF A sGC STIMULATOR AND AN sGC ACTIVATOR FOR CONDITIONS WHEREIN THE HEME GROUP OF sGC IS OXIDIZED OR WHEREIN sGC IS DEFICIENT IN HEME GUCY1A1, GUCY1B1, GUCY1A2 NPSR1 3795/4885AKR1C3 635/4885MAPT 4679/4885
US-20260000653-A1 TREATMENT OF CNS DISEASES WITH sGC STIMULATORS PDE9A, PDE2A, GUCY1A2 NPSR1 2001/4885AKR1C3 4147/4885MAPT 1030/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.