Oxalic Acid

Oxalic Acid

SCHEMBL8010108

Cn1nc(N2CCN(CCc3ccccc3)CC2)c2c1-c1ccccc1CC2.O=C(O)C(=O)O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.47
HRH4 Q9H3N8 5/20 0.47
HRH2 P25021 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
DRD4 P21917 1/20 0.43
DRD2 P14416 4/20 0.43
SIGMAR1 Q99720 4/20 0.43
HTR2A P28223 3/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 3/20 0.43
HTR1A P08908 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KCNH2 Q12809 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8011492 0.95 HRH1 (0.51) HRH1HRH4HRH2HRH3DRD4
SCHEMBL8015866 0.85 HTR1A (0.47) HRH1HRH4DRD2HTR1AMEN1
Oxalic Acid SCHEMBL8011549 0.84 HRH1 (0.46) HRH1HRH4HRH2HRH3DRD2
SCHEMBL8000858 0.83 DRD4 (0.47) HRH1HRH4HRH2HRH3DRD4
Oxalic Acid SCHEMBL8011723 0.80 DRD4 (0.67) HRH1HRH4HRH2HRH3DRD4
SCHEMBL8012631 0.78 HRH1 (0.49) HRH1HRH4HRH2HRH3DRD4
SCHEMBL8010100 0.75 KDR (0.49) DRD4DRD2SIGMAR1HTR2CHTR1A
SCHEMBL8008914 0.74 SMARCA2 (0.45) HRH1HRH4HRH2HRH3
SCHEMBL8009072 0.74 DRD4 (0.73) HRH1HRH4HRH2HRH3DRD4
SCHEMBL8008902 0.72 HRH1 (0.47) HRH1HRH4HRH2HRH3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080745-A Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands MERCK SHARP & DOHME LIMITED (GB) 2000-06-27 US disclosed
EP-0724572-B1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME (GB) 1998-12-16 EP disclosed
EP-0724572-A1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1996-08-07 EP disclosed
WO-1995007893-A1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1995-03-23 WO disclosed