SCHEMBL8010669

SCHEMBL8010669

Cc1cc(N2CCN(C(=O)COc3ccc4[nH]c(=O)oc4c3)CC2)ccc1I

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
ALDH1A1 P00352 4/20 0.54
MAPT P10636 3/20 0.54
GAA P10253 2/20 0.54
KMT2A Q03164 2/20 0.49
KCNH2 Q12809 1/20 0.48
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
RECQL P46063 1/20 0.45
MEN1 O00255 1/20 0.45
MAPK1 P28482 1/20 0.43
HTR1A P08908 1/20 0.43
HTR1D P28221 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016624 0.84 GRIN1 (0.55) KDM4EALDH1A1MAPTGAAKCNH2
SCHEMBL2017436 0.84 KCNH2 (0.52) KDM4EALDH1A1MAPTGAAKCNH2
SCHEMBL2017504 0.84 KCNH2 (0.66) KDM4EALDH1A1MAPTGAAKCNH2
SCHEMBL8010801 0.77 DRD2 (0.48) KDM4EALDH1A1MAPTGAAKMT2A
SCHEMBL2022608 0.75 KCNH2 (0.53) MAPTGAAKCNH2
SCHEMBL2015494 0.75 KCNH2 (0.51) MAPTGAAKCNH2
SCHEMBL2018259 0.75 KCNH2 (0.64) KDM4EMAPTGAAKCNH2
SCHEMBL8012931 0.72 MEN1 (0.55) KDM4EALDH1A1MAPTGAAKMT2A
SCHEMBL23123753 0.71 HTR1A (0.50) KDM4EALDH1A1KCNH2HTR1A
SCHEMBL12232768 0.71 ACHE (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137843-A2 NMDA RECEPTOR ANTAGONISTS FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS EMORY UNIVERSITY (US) 2009-11-12 WO disclosed
WO-2009006437-A1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION EMORY UNIVERSITY (US) 2009-01-08 WO disclosed