SCHEMBL8011007

SCHEMBL8011007

Cc1c(CO)ncn1C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12344479 0.79
SCHEMBL17689166 0.77
SCHEMBL12569981 0.77 ALDH1A1 (0.32)
SCHEMBL8011000 0.76
SCHEMBL859688 0.76
SCHEMBL22125858 0.76
SCHEMBL25868933 0.76
SCHEMBL5655389 0.75 ADORA2A (0.38)
SCHEMBL21486293 0.74 APOBEC3A (0.33)
SCHEMBL13384272 0.74 KDM4E (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219970-A1 DIHYDROCHROMENE DERIVATIVES Sumitomo Pharma Co., Ltd. (JP) 2023-07-13 US disclosed
US-11639357-B2 Dihydrochromene derivatives Sumitomo Pharma Co., Ltd. (JP) 2023-05-02 US disclosed
US-20210002290-A1 DIHYDROCHROMENE DERIVATIVES SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-01-07 US disclosed
US-10807993-B2 Dihydrochromene derivatives SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-10-20 US disclosed
US-20200216461-A1 DIHYDROCHROMENE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-07-09 US disclosed
US-9315521-B2 Pyrimidines as novel therapeutic agents UNIVERSITé LAVAL (CA) 2016-04-19 US disclosed
US-9315521-B2 Pyrimidines as novel therapeutic agents UNIVERSITé LAVAL (CA) 2016-04-19 US disclosed
US-6107312-A BACTERICIDE BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-08-22 US disclosed
EP-0683776-B1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-07 EP disclosed
US-5587389-A Substituted heteroarylaklylthiopyridines for controlling helicobacter bacteria BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-12-24 US disclosed
WO-1996000224-A1 4-S- AND N-SUBSTITUTED 6-ALKYLPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-01-04 WO disclosed
US-4292431-A Process for the production of hydroxymethylimidazoles KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 1981-09-29 US disclosed