SCHEMBL8013307

SCHEMBL8013307

COc1ccc2c(c1)N(C(=O)OC(C)(C)C)CCC2O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
STS P08842 2/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
EPHX2 P34913 1/20 0.42
KDM1A O60341 1/20 0.42
HTT P42858 2/20 0.42
GPR119 Q8TDV5 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TGFBR1 P36897 2/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CRHBP P24387 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649609 0.89 ALDH1A1 (0.48) ALDH1A1STSMEN1KMT2AEPHX2
SCHEMBL6649701 0.86 ALDH1A1 (0.43) ALDH1A1STSMEN1KMT2AEPHX2
SCHEMBL6650959 0.86 ALDH1A1 (0.43) ALDH1A1STSMEN1KMT2AEPHX2
SCHEMBL8878468 0.86 ALDH1A1 (0.43) ALDH1A1STSMEN1KMT2AEPHX2
SCHEMBL8878473 0.86 ALDH1A1 (0.43) ALDH1A1STSMEN1KMT2AEPHX2
SCHEMBL19892893 0.84 ALDH1A1 (0.44) ALDH1A1STSMEN1KMT2AKDM1A
SCHEMBL31064582 0.81 GPR119 (0.43) ALDH1A1STSMEN1KMT2AKDM1A
SCHEMBL29457639 0.80 KDM1A (0.55) MEN1KMT2AKDM1AGPR119KDM4E
SCHEMBL2174623 0.80 KDM1A (0.55) MEN1KMT2AKDM1AGPR119KDM4E
SCHEMBL29457605 0.80 KDM1A (0.55) MEN1KMT2AKDM1AGPR119KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6093821-A MAKING 6-(PHENYL OR HETEROARYL)-1,2-DIHYDRO-N-1-PROTECTED QUINOLINE BY REACTING THE CORRESPONDING 6-HALO-DERIVATIVE WITH AN ORGANOBORATE AND ACID TREATMENT TO FORM THE 6-BORO-DERIVATIVE, COUPLING WITH PHENYL OR HETEROARYL HALIDE LIGAND PHARMACEUTICALS INCORPORATED (US) 2000-07-25 US disclosed