SCHEMBL8015015

SCHEMBL8015015

Cc1[nH]c(C)c2c(=O)[nH]nc(Cc3cccc(C=O)c3)c12

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.43
AR P10275 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
DAO P14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76940 0.82 PARP1 (0.57) PARP1ARALDH1A1CYP2C9HPGD
SCHEMBL76810 0.80 PARP1 (0.48) PARP1
SCHEMBL13265573 0.77 PARP1 (0.71) PARP1ARCYP2C9
SCHEMBL5096925 0.74 PARP1 (0.70) PARP1
SCHEMBL13665692 0.71 MEN1 (0.52) AR
SCHEMBL13776979 0.71 PARP1 (0.65) PARP1
SCHEMBL4435003 0.68 PARP1 (0.67) PARP1
SCHEMBL6852425 0.68 ALDH1A1 (0.52) ALDH1A1
SCHEMBL20546828 0.66 MAOA (0.59) ALDH1A1DAO
SCHEMBL20546750 0.66 MAOA (0.62) ALDH1A1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093032-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA AB (SE) 2009-07-30 WO disclosed