SCHEMBL8015244

SCHEMBL8015244

O=C(NN1CCN(OC(F)(F)F)CC1C(=O)c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.40
POLB P06746 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 2/20 0.38
SLC6A12 P48065 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
MCHR1 Q99705 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972859 0.69 HSD11B1 (0.49) HSD11B1CYP2D6
SCHEMBL2218785 0.69 HTT (0.51) CYP3A4CYP2C9CYP2C19
SCHEMBL7972582 0.67 MAPT (0.43) ALDH1A1CYP2D6NPC1RAB9ASMN1; SMN2
SCHEMBL7972577 0.62 CYP2D6 (0.59) HSD11B1POLBCYP2D6CYP2C9CYP2C19
SCHEMBL2400667 0.62 HTT (0.53) ALDH1A1SMN1; SMN2
SCHEMBL27695426 0.62 HTT (0.53) ALDH1A1SMN1; SMN2
SCHEMBL9185373 0.62 CYP2D6 (0.62) HSD11B1ALDH1A1CYP2D6
SCHEMBL28006890 0.61 NPC1 (0.66) POLBALDH1A1CYP2C9NPC1RAB9A
SCHEMBL8419841 0.61 CYP2D6 (0.47) HSD11B1POLBALDH1A1CYP2D6CYP1A2
SCHEMBL28694284 0.60 KDM4E (0.47) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968201-A2 NEW AMINOPIPERAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-01-05 EP disclosed
WO-1998035951-A2 NEW AMINOPIPERAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-20 WO disclosed