SCHEMBL8015367

SCHEMBL8015367

Cc1ccc(CN(C)C)s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT6 Q96LA8 1/20 0.50
RIPK1 Q13546 1/20 0.50
CYP2A6 P11509 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
THRB P10828 2/20 0.41
TP53 P04637 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.40
ADRA1D P25100 2/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HRH3 Q9Y5N1 1/20 0.36
TSHR P16473 1/20 0.36
EED O75530 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10154745 0.80 RIPK1 (0.50) PRMT6RIPK1CYP2A6CYP2D6CYP2C19
SCHEMBL12203994 0.77 RIPK1 (0.47) PRMT6RIPK1THRBTP53TRPM8
SCHEMBL18355118 0.77 RIPK1 (0.44) PRMT6RIPK1THRBTP53TRPM8
SCHEMBL13185588 0.76 CYP2A6 (0.44) RIPK1CYP2A6CYP2D6CYP2C19TP53
SCHEMBL10151102 0.76 RIPK1 (0.43) PRMT6RIPK1THRBTP53TRPM8
SCHEMBL7277336 0.74 CYP2A6 (0.43) RIPK1CYP2A6CYP2D6CYP2C19THRB
SCHEMBL8015366 0.74 CYP2A6 (0.43) RIPK1CYP2A6CYP2D6CYP2C19ALDH1A1
SCHEMBL21127888 0.74 CYP2A6 (0.43) RIPK1CYP2A6CYP2D6CYP2C19ALDH1A1
SCHEMBL8008762 0.74 CYP2A6 (0.43) RIPK1CYP2A6CYP2D6CYP2C19ALDH1A1
SCHEMBL621621 0.74 CYP2A6 (0.43) CYP2A6CYP2D6CYP2C19ADRA1DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230339943-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVES Guangdong Raynovent Biotech Co., Ltd. (CN) 2023-10-26 US disclosed
US-20230339943-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVES Guangdong Raynovent Biotech Co., Ltd. (CN) 2023-10-26 US disclosed
US-11725009-B2 Anti-influenza virus pyrimidine derivative Guangdong Raynovent Biotech Co., Ltd. (CN) 2023-08-15 US disclosed
US-11725009-B2 Anti-influenza virus pyrimidine derivative Guangdong Raynovent Biotech Co., Ltd. (CN) 2023-08-15 US disclosed
US-20220135558-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVE Guangdong Raynovent Biotech Co., Ltd. (CN) 2022-05-05 US disclosed
US-11136319-B2 Anti-influenza virus pyrimidine derivative Guangdong Raynovent Biotech Co., Ltd. (CN) 2021-10-05 US disclosed
US-20210032238-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVE Guangdong Raynovent Biotech Co., Ltd. (CN) 2021-02-04 US disclosed
EP-3502112-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVE Guangdong Raynovent Biotech Co., Ltd. (CN) 2019-06-26 EP disclosed
US-8034949-B2 Pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-10-11 US disclosed
US-8034949-B2 Pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-10-11 US disclosed
US-6107312-A BACTERICIDE BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-08-22 US disclosed
EP-0683776-B1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-07 EP disclosed
CN-1155284-A Thipyridines for use in control of helicobacter bacteria BYK GULDEN LOMBERG CHEM FAB (DE) 1997-07-23 CN disclosed
EP-0764160-A1 THIOPYRIDINES FOR USE IN THE CONTROL OF HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1997-03-26 EP disclosed
US-5587389-A Substituted heteroarylaklylthiopyridines for controlling helicobacter bacteria BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-12-24 US disclosed
WO-1996000224-A1 4-S- AND N-SUBSTITUTED 6-ALKYLPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-01-04 WO disclosed
WO-1995034553-A1 THIOPYRIDINES FOR USE IN THE CONTROL OF HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1995-12-21 WO disclosed
EP-0683776-A1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1995-11-29 EP disclosed
WO-1994019346-A1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-09-01 WO disclosed
EP-0177016-B1 PYRIDYLOXY DERIVATIVES Ikeda Mohando Co., Ltd. (JP) 1993-06-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11725009-B2 Anti-influenza virus pyrimidine derivative ENTPD5, NUDT15, ITPA PRMT6 2345/4885RIPK1 3676/4885CYP2A6 1305/4885
US-20220135558-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVE ENTPD5, NUDT15, ITPA PRMT6 2345/4885RIPK1 3676/4885CYP2A6 1305/4885
US-20230339943-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVES ENTPD5, NUDT1, ITPA PRMT6 2248/4885RIPK1 3574/4885CYP2A6 1284/4885
US-20210032238-A1 ANTI-INFLUENZA VIRUS PYRIMIDINE DERIVATIVE ENTPD5, NUDT15, ITPA PRMT6 2345/4885RIPK1 3676/4885CYP2A6 1305/4885
US-11136319-B2 Anti-influenza virus pyrimidine derivative ENTPD5, NUDT15, ITPA PRMT6 2345/4885RIPK1 3676/4885CYP2A6 1305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.