SCHEMBL8016752

SCHEMBL8016752

NS(=O)(=O)c1cc(Br)cc(C(F)(F)F)c1.Nc1cc(Br)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.43
CA1 P00915 9/20 0.43
CA9 Q16790 9/20 0.43
CA3 P07451 1/20 0.43
KIF11 P52732 2/20 0.41
NOTUM Q6P988 1/20 0.40
CA12 O43570 3/20 0.38
CA5A P35218 4/20 0.38
CNR1 P21554 1/20 0.38
ACP1 P24666 1/20 0.38
CA4 P22748 2/20 0.37
CA6 P23280 2/20 0.37
CA7 P43166 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA5B Q9Y2D0 2/20 0.37
PLA2G1B P04054 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
APEX1 P27695 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4807857 0.92 KIF11 (0.47) CA2CA1CA9CA3KIF11
SCHEMBL134690 0.82 TSHR (0.46) CA2CA1CA9KIF11NOTUM
SCHEMBL29426986 0.82 TSHR (0.46) CA2CA1CA9KIF11NOTUM
SCHEMBL2920504 0.78 KIF11 (0.55) CA2CA1CA9CA3KIF11
SCHEMBL11292063 0.74 ACP1 (0.49) CA2CA1CA9NOTUMCA5A
SCHEMBL700367 0.74 NOTUM (0.45) CA2CA1CA9NOTUMCA5A
SCHEMBL12098234 0.74 NOTUM (0.49) CA2CA1CA9KIF11NOTUM
SCHEMBL30253146 0.74 NOTUM (0.49) CA2CA1CA9KIF11NOTUM
SCHEMBL2810521 0.73 LMNA (0.42) CA2CA1CA9KIF11CA12
SCHEMBL13277683 0.73 ACP1 (0.48) CA2CA1CA9NOTUMCA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971892-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Astra Pharmaceuticals Limited (GB) 2000-01-19 EP disclosed
WO-1998042670-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRA PHARMACEUTICALS LTD. (GB) 1998-10-01 WO disclosed