SCHEMBL8017003

SCHEMBL8017003

CC(C)c1ccc(S(=O)(=O)c2nnn3c2nc(N2CCSCC2)c2sccc23)cc1

nearest known ligand 0.84

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.84
RXFP1 Q9HBX9 10/20 0.73
HTR6 P50406 4/20 0.67
MAPT P10636 4/20 0.63
ALDH1A1 P00352 1/20 0.60
HPGD P15428 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029215 0.90 RXFP1 (0.82) THRBRXFP1HTR6MAPT
SCHEMBL8027286 0.87 THRB (0.81) THRBRXFP1HTR6MAPTALDH1A1
SCHEMBL8030781 0.82 RXFP1 (0.85) THRBRXFP1HTR6MAPT
SCHEMBL8019324 0.80 RXFP1 (1.00) THRBRXFP1HTR6MAPT
SCHEMBL8016821 0.80 HTR6 (0.85) RXFP1HTR6MAPT
SCHEMBL8028230 0.79 HTR6 (0.98) THRBRXFP1HTR6
SCHEMBL8018275 0.79 RXFP1 (0.82) THRBRXFP1HTR6MAPT
SCHEMBL8028237 0.79 HTR6 (0.85) RXFP1HTR6MAPT
SCHEMBL8026961 0.77 RXFP1 (1.00) THRBRXFP1HTR6MAPT
SCHEMBL8019326 0.77 HTR6 (0.98) THRBRXFP1HTR6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed