SCHEMBL8017249

SCHEMBL8017249

COc1cccc(OC)c1C1C[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CCC[C@@]4(C)CC[C@@H]32)NC1=O

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 3/20 0.38
MBOAT4 Q96T53 3/20 0.36
GRIN1 Q05586 4/20 0.36
GRIN2B Q13224 4/20 0.36
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
NR1I3 Q14994 1/20 0.35
CYP19A1 P11511 3/20 0.35
AR P10275 1/20 0.33
SRD5A2 P31213 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8023088 0.90 SRD5A1 (0.39) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8006579 0.85 DDB1 (0.46) SRD5A1MBOAT4CYP19A1
SCHEMBL8017204 0.84 MBOAT4 (0.38) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8023121 0.84 DDB1 (0.42) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8016699 0.82 SRD5A1 (0.49) SRD5A1ARSRD5A2
SCHEMBL8710564 0.81 MBOAT4 (0.38) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8019115 0.80 SRD5A1 (0.37) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8019044 0.79 MBOAT4 (0.35) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8020709 0.78 MBOAT4 (0.35) SRD5A1MBOAT4GRIN1GRIN2BCDK5
SCHEMBL8020694 0.78 MBOAT4 (0.36) SRD5A1MBOAT4GRIN1GRIN2BCDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed