SCHEMBL8023121

SCHEMBL8023121

COc1ccc(C2C[C@@]3(C)[C@@H](CC[C@H]4[C@@H]5CCC[C@@]5(C)CC[C@@H]43)NC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
SRD5A1 P18405 2/20 0.39
CYP19A1 P11511 6/20 0.37
MBOAT4 Q96T53 3/20 0.36
MMP1 P03956 1/20 0.36
MMP13 P45452 1/20 0.36
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
NR1I3 Q14994 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710564 0.89 MBOAT4 (0.38) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8006579 0.89 DDB1 (0.46) DDB1CRBNSRD5A1CYP19A1MBOAT4
SCHEMBL8020694 0.86 MBOAT4 (0.36) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8017204 0.84 MBOAT4 (0.38) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8017249 0.84 SRD5A1 (0.38) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8023088 0.82 SRD5A1 (0.39) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8018769 0.79 SRD5A1 (0.41) DDB1CRBNSRD5A1CYP19A1MBOAT4
SCHEMBL8019044 0.79 MBOAT4 (0.35) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL8019115 0.78 SRD5A1 (0.37) SRD5A1CYP19A1MBOAT4CDK5CDK5R1
SCHEMBL9546857 0.77 CDK5 (0.43) SRD5A1CYP19A1MBOAT4CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed