SCHEMBL8006579

SCHEMBL8006579

COc1cccc(C2C[C@@]3(C)[C@@H](CC[C@H]4[C@@H]5CCC[C@@]5(C)CC[C@@H]43)NC2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.46
CRBN Q96SW2 1/20 0.46
SRD5A1 P18405 2/20 0.41
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR2C P28335 2/20 0.35
CYP19A1 P11511 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GID4 Q8IVV7 1/20 0.35
MBOAT4 Q96T53 2/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
ALOX12 P18054 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8023121 0.89 DDB1 (0.42) DDB1CRBNSRD5A1CYP19A1MBOAT4
SCHEMBL8019044 0.85 MBOAT4 (0.35) SRD5A1CYP19A1MBOAT4
SCHEMBL8017249 0.85 SRD5A1 (0.38) SRD5A1CYP19A1MBOAT4
SCHEMBL8017204 0.83 MBOAT4 (0.38) SRD5A1KMT2ACYP19A1MBOAT4LMNA
SCHEMBL8710564 0.81 MBOAT4 (0.38) SRD5A1CYP19A1MBOAT4
SCHEMBL8023088 0.81 SRD5A1 (0.39) SRD5A1CYP19A1MBOAT4ALDH1A1LMNA
SCHEMBL8024003 0.81 DDB1 (0.41) DDB1CRBNSRD5A1MEN1NPC1
SCHEMBL8020694 0.79 MBOAT4 (0.36) SRD5A1CYP19A1MBOAT4
SCHEMBL8020709 0.77 MBOAT4 (0.35) SRD5A1CYP19A1MBOAT4
SCHEMBL8019115 0.77 SRD5A1 (0.37) SRD5A1CYP19A1MBOAT4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed