SCHEMBL8017285

SCHEMBL8017285

CCOC(=O)[C@H](CC(C)C)NCCNC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.46
CTSL P07711 2/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
MAPT P10636 1/20 0.42
POLB P06746 1/20 0.41
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
PPID Q08752 1/20 0.39
CA12 O43570 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460122 0.88 CTSL (0.48) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL14280789 0.84 MEN1 (0.48) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL8977043 0.84 MEN1 (0.54) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL8976845 0.83 CAPN1 (0.47) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL15374288 0.82 CYP1A2 (0.59) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL15107084 0.82 CYP1A2 (0.59) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL9596442 0.82 CYP1A2 (0.59) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL8017762 0.81 CYP1A2 (0.49) CAPN1CTSLCTSBCTSSCTSK
Hydrochloric Acid SCHEMBL30231858 0.80 CAPN1 (0.46) CAPN1CTSLCTSBCTSSCTSK
SCHEMBL10743743 0.78 PPID (0.43) CAPN1CTSLCTSBKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706532-B1 Peptides having endothelin antagonictic activity,their preparation and pharmaceutical compositions FUJISAWA PHARMACEUTICAL CO (JP) 2000-02-02 EP disclosed
EP-0706532-A1 NEW COMPOUND AND ITS PREPARATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-17 EP disclosed
WO-1995000537-A1 NEW COMPOUND AND ITS PREPARATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-01-05 WO disclosed