SCHEMBL8017451

SCHEMBL8017451

COC(=O)CCc1cc2ccc(C(=O)O)cc2n1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 2/20 0.40
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
HCAR3 P49019 1/20 0.36
MCL1 Q07820 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA7 P43166 1/20 0.36
TPMT P51580 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PDE2A O00408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9105728 0.81 NPC1 (0.53) MTNR1AMTNR1BNPC1RAB9ACYP11B1
SCHEMBL10983071 0.77 OXER1 (0.47) HCAR3ALDH1A1
SCHEMBL7422778 0.74 KDM4E (0.40) MTNR1AMTNR1BKDM4ECYP11B1CYP11B2
SCHEMBL29703917 0.74 HDAC6 (0.50) NPC1RAB9AHCAR3ALDH1A1
SCHEMBL16413519 0.73 L3MBTL1 (0.56) MTNR1AMTNR1BKDM4EMCL1ALDH1A1
SCHEMBL17680280 0.72 MTNR1A (0.46) MTNR1AMTNR1BNPC1RAB9AKDM4E
SCHEMBL31721264 0.70 KDM4E (0.46) KDM4EHCAR3MCL1ALDH1A1CA12
SCHEMBL13290538 0.70 KDM4E (0.46) KDM4EHCAR3MCL1ALDH1A1
SCHEMBL28269380 0.69 KDM4E (0.45) RAB9AKDM4EHCAR3MCL1ALDH1A1
SCHEMBL28271125 0.69 KDM4E (0.45) KDM4EHCAR3MCL1ALDH1A1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069156-A Indole derivatives as cGMP-PDE inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-05-30 US disclosed