SCHEMBL8018877

SCHEMBL8018877

O=C(O)c1ccc(S(=O)(=O)Nc2cccc(B(O)O)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.62
PFKFB3 Q16875 1/20 0.54
CA12 O43570 2/20 0.54
CA9 Q16790 2/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
KMT2A Q03164 6/20 0.53
MEN1 O00255 4/20 0.53
MAPT P10636 1/20 0.51
ALDH1A1 P00352 1/20 0.51
ITGA1 P56199 2/20 0.50
AKR1C3 P42330 1/20 0.50
GAA P10253 1/20 0.50
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
THRB P10828 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8013313 0.97 POLB (0.59) POLBPFKFB3CA12CA9CA1
SCHEMBL1687192 0.97 POLB (0.59) POLBPFKFB3CA12CA9CA1
SCHEMBL8009397 0.87 KMT2A (0.65) PFKFB3KMT2AMEN1MAPTTHRB
SCHEMBL15649873 0.84 HSD17B2 (0.56) POLBCA1CA2KMT2AMEN1
SCHEMBL7997931 0.83 HTR6 (0.68) POLBCA9CA1CA2KMT2A
SCHEMBL28632297 0.83 L3MBTL1 (0.58) CA1CA2KMT2AMEN1MAPT
SCHEMBL12260987 0.83 CA12 (0.59) CA12CA9CA1CA2KMT2A
SCHEMBL3715141 0.80 CA12 (0.75) POLBCA12CA9CA1CA2
SCHEMBL22653513 0.80 POLB (0.65) POLBPFKFB3CA12CA9CA1
SCHEMBL664321 0.80 KMT2A (0.75) POLBCA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000035904-A1 INHIBITORS OF β-LACTAMASES AND USES THEREFOR NORTHWESTERN UNIVERSITY (US) 2000-06-22 WO disclosed