SCHEMBL8018891

SCHEMBL8018891

CC(C)(C)OC(=O)NC1(C(=O)O)CC1C(=O)c1cccc(Br)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
BCL2 P10415 1/20 0.36
BECN1 Q14457 1/20 0.36
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
TP53BP1 Q12888 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8018983 0.87 L3MBTL1 (0.39) MEN1KMT2ACTSSCTSKALDH1A1
SCHEMBL8025163 0.87 SIRT2 (0.40) SMN1; SMN2MEN1KMT2AALDH1A1CYP2C19
SCHEMBL8022535 0.81 CYP2C19 (0.52) SMN1; SMN2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8025263 0.81 DPP8 (0.37) MEN1KMT2ARAB9AMAPT
SCHEMBL8025124 0.73 SMN1; SMN2 (0.41) SMN1; SMN2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8020026 0.72 BACE1 (0.38) SMN1; SMN2MEN1KMT2AALDH1A1NPC1
SCHEMBL27805616 0.72 KDM1A (0.38) SMN1; SMN2CTSBCTSSCTSKBCL2
SCHEMBL2075585 0.72 MAPK1 (0.46) SMN1; SMN2MEN1KMT2ACTSSCTSK
SCHEMBL27512707 0.70 BACE1 (0.37) SMN1; SMN2MEN1KMT2AALDH1A1NPC1
SCHEMBL15767766 0.70 KDM1A (0.46) SMN1; SMN2CTSBCTSSCTSKBCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973720-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.p.A. (IT) 2000-01-26 EP disclosed
WO-1998040344-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 1998-09-17 WO disclosed