SCHEMBL8022535

SCHEMBL8022535

O=C(NC1(C(=O)O)CC1C(=O)c1cccc(Br)c1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.52
MAPK1 P28482 1/20 0.52
SMN1; SMN2 Q16637 5/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 2/20 0.44
FAAH O00519 1/20 0.43
KMT2A Q03164 7/20 0.42
ALDH1A1 P00352 6/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 6/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
MAPT P10636 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8020166 0.85 MAPK1 (0.52) CYP2C19MAPK1SMN1; SMN2NPC1RAB9A
SCHEMBL8018575 0.85 MAPK1 (0.52) CYP2C19MAPK1SMN1; SMN2NPC1RAB9A
SCHEMBL8018891 0.81 SMN1; SMN2 (0.38) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL8017815 0.74 PARP1 (0.47) CYP2C19SMN1; SMN2KMT2AALDH1A1GAA
SCHEMBL8025124 0.71 SMN1; SMN2 (0.41) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL1740252 0.70 MAPK1 (0.60) CYP2C19MAPK1FAAHKMT2AALDH1A1
SCHEMBL4652925 0.69 SMN1; SMN2 (0.71) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL17336679 0.69 SMN1; SMN2 (0.64) CYP2C19SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL7417055 0.69 MAPK1 (1.00) CYP2C19MAPK1FAAHKMT2AALDH1A1
SCHEMBL27536880 0.68 PARP1 (0.43) CYP2C19MAPK1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973720-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.p.A. (IT) 2000-01-26 EP disclosed
WO-1998040344-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 1998-09-17 WO disclosed