SCHEMBL8018987

SCHEMBL8018987

Bc1cc(CN)ccc1C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.39
LOXL2 Q9Y4K0 3/20 0.37
ABAT P80404 1/20 0.36
PNMT P11086 1/20 0.35
ENPP2 Q13822 1/20 0.35
ST14 Q9Y5Y6 1/20 0.35
CYP2A6 P11509 1/20 0.35
CSNK2A1 P68400 3/20 0.35
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
LOX P28300 1/20 0.34
TAAR1 Q96RJ0 2/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PSIP1 O75475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13772758 0.79 TRPA1 (0.43) CYP2A6GAAPKMTAAR1NOS3
SCHEMBL29406921 0.78 ALDH1A1 (0.46) HRH3LOXL2ABATPNMTENPP2
SCHEMBL39710 0.78 ALDH1A1 (0.46) HRH3LOXL2ABATPNMTENPP2
SCHEMBL14216527 0.77 CYP4F2 (0.35)
Iodide SCHEMBL31233435 0.76 ALDH1A1 (0.44) HRH3LOXL2ABATPNMTENPP2
SCHEMBL13772884 0.76 CNR1 (0.45)
SCHEMBL14407078 0.76 ESR1 (0.48) GAA
SCHEMBL21699644 0.74 HRH3 (0.40) HRH3LOXL2ABATPNMTENPP2
SCHEMBL2221947 0.74 TAAR1 (0.43) HRH3LOXL2ABATPNMTENPP2
SCHEMBL8211010 0.74 ALDH1A1 (0.52) HRH3LOXL2ABATGAANOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100167-A1 DUAL PHARMACOPHORES-PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed
WO-2009100166-A1 DUAL PHARMACOPHORES-PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed