SCHEMBL8019014

SCHEMBL8019014

N#CC(O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.75
ACP3 P15309 2/20 0.44
PTGS2 P35354 1/20 0.44
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
MMP3 P08254 1/20 0.41
BCL2L1 Q07817 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
TRPA1 O75762 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PGR P06401 1/20 0.39
FFAR1 O14842 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21114421 0.86 TSHR (1.00) TSHRTRPA1ALDH1A1
SCHEMBL196731 0.86 TSHR (1.00) TSHRTRPA1ALDH1A1
SCHEMBL6061809 0.86 TSHR (1.00) TSHRTRPA1ALDH1A1
SCHEMBL1820543 0.86 TSHR (1.00) TSHRTRPA1ALDH1A1
SCHEMBL11161987 0.82 TSHR (0.67) TSHRCTSSCTSKTRPA1CA2
SCHEMBL10566017 0.82 TSHR (0.67) TSHRCTSSCTSKTRPA1CA2
SCHEMBL6056000 0.81 TSHR (0.79) TSHRMMP3BCL2L1TRPA1CYP3A4
SCHEMBL6390318 0.78 PTGS2 (0.48) TSHRACP3PTGS2CHRNB2CHRNA4
SCHEMBL8019224 0.78 TSHR (0.67) TSHRCA1CA2
SCHEMBL11675463 0.77 CHRNB2 (0.45) TSHRACP3PTGS2CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111072586-B N-hydroxy-3-substituted-5-carboxamide compound, preparation method and application thereof 中国药科大学 2023-06-09 CN disclosed
EP-0711836-B1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide MITSUBISHI RAYON CO (JP) 2000-02-02 EP disclosed
US-5736385-A NITRILASE OR NITRILE HYDRATASE HYDROLYSIS OF A CYANOHYDRIN WHILE AUTOMATICALLY CONTROLLING CYANOHYDRIN CONCENTRATION NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
EP-0711836-A1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-05-15 EP disclosed