SCHEMBL8021079

SCHEMBL8021079

COc1cc2c(cc1OC)C(c1ccccc1F)=NCC2

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.71
RAD52 P43351 1/20 0.71
MAPK10 P53779 9/20 0.60
MAPK14 Q16539 2/20 0.60
LMNA P02545 3/20 0.59
MAPT P10636 3/20 0.59
NPSR1 Q6W5P4 2/20 0.59
HTT P42858 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
ALDH1A1 P00352 3/20 0.59
KDM4E B2RXH2 3/20 0.54
GAA P10253 1/20 0.54
MAOA P21397 1/20 0.54
GLA P06280 1/20 0.52
RCE1 Q9Y256 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704178 0.86 MAPK10 (0.61) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL17144905 0.82 ALDH1A1 (0.71) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL5355121 0.81 MAPK10 (0.80) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL30979840 0.81 MAPK10 (0.80) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL10333535 0.81 PKM (0.68) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL13478295 0.78 PKM (0.64) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL10425807 0.77 PKM (0.63) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL28224519 0.76 ALDH1A1 (0.72) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL31011321 0.75 ALDH1A1 (0.76) PKMRAD52MAPK10MAPK14LMNA
SCHEMBL28180887 0.75 ALDH1A1 (0.76) PKMRAD52MAPK10MAPK14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000044725-A1 FUSED DIHYDROPYRIDINES AND USE OF FUSED DIHYDROPYRIDINES IN THE PREPARATION OF AGENTS FOR THE TREATMENT OF EPILEPSY BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-08-03 WO disclosed
WO-1992011242-A1 FUNGICIDAL ISOQUINOLINE DERIVATIVES SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1992-07-09 WO disclosed
EP-0491441-A1 Fungicidal isoquinoline derivatives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1992-06-24 EP disclosed