SCHEMBL8021114

SCHEMBL8021114

CC(C)(C)C1(Cc2ccccc2Cl)CO1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.38
PNMT P11086 1/20 0.38
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TAAR1 Q96RJ0 3/20 0.37
CYP2A13 Q16696 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HSD11B1 P28845 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
AOC3 Q16853 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ATM Q13315 1/20 0.35
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2126992 0.81 TAAR1 (0.40) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL2127284 0.79 SLC6A2 (0.36) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL16165985 0.78 CNR2 (0.35) KDM4E
SCHEMBL16165982 0.78 GAA (0.33) KDM4EAOC3
SCHEMBL9353042 0.72 KCNH2 (0.39) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL29290780 0.71 IDO1 (0.41) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL31142998 0.69 IDO1 (0.38) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL6573590 0.69 IDO1 (0.38) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL9683385 0.69 ALDH1A1 (0.40) IDO1PNMTHTTKDM4ETAAR1
SCHEMBL1282488 0.68 L3MBTL1 (0.48) NPC1RAB9AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618918-B1 PROCESS FOR THE PREPARATION OF ETHER SOLUTIONS OF GRIGNARD COMPOUNDS ZENECA LTD (GB) 2000-01-19 EP disclosed
EP-0594658-B1 PROCESS FOR THE PREPARATION OF ARYL AND ARALKYL MAGNESIUM HALIDES ZENECA LTD (GB) 1996-11-20 EP disclosed
EP-0594658-A1 PROCESS FOR THE PREPARATION OF ARYL AND ARALKYL MAGNESIUM HALIDES. ZENECA LTD (GB) 1994-05-04 EP disclosed
US-5242625-A Preparation of Grignard reagents in high boiling solvent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-07 US disclosed
US-5209459-A Alternative ether solvent for preparation of arylmagnesium halide Grignard reagent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-11 US disclosed
WO-1993002086-A1 PROCESS FOR THE PREPARATION OF ARYL AND ARALKYL MAGNESIUM HALIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-04 WO disclosed