SCHEMBL8021469

SCHEMBL8021469

CC(C)c1cc2c(c(C(C)C)c1O)CCC(C)(COc1ccc(CC3SC(=O)NC3=O)cc1)O2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
MAPT P10636 2/20 0.51
KMT2A Q03164 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
ALDH1A1 P00352 1/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
HPGD P15428 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
HSD17B10 Q99714 1/20 0.51
THRA P10827 2/20 0.44
THRB P10828 2/20 0.44
PPARG P37231 8/20 0.42
FFAR1 O14842 7/20 0.41
PPARA Q07869 4/20 0.41
HRH3 Q9Y5N1 1/20 0.40
MPC2 O95563 1/20 0.40
CYP2C8 P10632 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10639426 0.93 MEN1 (0.43) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10969847 0.87 CYP3A4 (0.43) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10640256 0.85 MEN1 (0.49) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10639191 0.85 MEN1 (0.52) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10639005 0.83 MEN1 (0.54) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10636378 0.82 MEN1 (0.40) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL7455277 0.81 ALDH1A1 (0.56) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10639049 0.79 CYP3A4 (0.56) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10640431 0.79 MEN1 (0.41) MEN1MAPTKMT2ATDP1ALDH1A1
SCHEMBL10641884 0.79 MEN1 (0.50) MEN1MAPTKMT2ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6110951-A LOWERING INSULIN DRUG THERAPY IN NON-OBESE, NON-DIABETIC INDIVIDUALS BETHESDA PHARMACEUTICALS, INC. 2000-08-29 US disclosed
US-5594015-A Thiazolidine derivatives for the treatment of psoriasis REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-01-14 US disclosed
US-5053420-A Antidiabetic agents KURTZ, THEODORE W. 1991-10-01 US disclosed
WO-1991005538-A2 THIAZOLIDINE DERIVATIVES FOR THE TREATMENT OF HYPERTENSION PERSHADSINGH HARRIHAR A (US) 1991-05-02 WO disclosed
EP-0139421-B1 THIAZOLIDINE DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1988-04-27 EP disclosed
US-4572912-A Thiazolidine derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1986-02-25 US disclosed
EP-0139421-A1 Thiazolidine derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1985-05-02 EP disclosed