SCHEMBL8022341

SCHEMBL8022341

COc1cc(Cl)c(C(=O)N(C)C(=O)N(C)Cc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
RAF1 P04049 2/20 0.49
MAP2K1 Q02750 2/20 0.49
HPGD P15428 2/20 0.46
GAA P10253 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
SRD5A1 P18405 1/20 0.46
SRD5A2 P31213 1/20 0.46
EGFR P00533 1/20 0.45
CTSV O60911 1/20 0.45
CTSL P07711 1/20 0.45
HTT P42858 1/20 0.45
HSP90AA1 P07900 1/20 0.45
APP P05067 2/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034161 0.92 APP (0.47) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8035939 0.89 RAF1 (0.44) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8031650 0.87 MEN1 (0.46) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8022338 0.85 TRPM8 (0.46) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8039011 0.85 HSP90AA1 (0.53) MEN1KMT2AHPGDGAARXFP1
SCHEMBL8034163 0.85 CTSV (0.47) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8035938 0.83 SRD5A1 (0.47) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8038345 0.82 HPGD (0.52) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8032086 0.81 NPC1 (0.47) MEN1KMT2ARAF1MAP2K1HPGD
SCHEMBL8041162 0.81 CTSV (0.60) HPGDSRD5A1SRD5A2CTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed