SCHEMBL8023948

SCHEMBL8023948

COc1cc(Cl)c(C(=O)NC(=O)NCC(F)(F)F)cc1O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PYGL P06737 13/20 0.46
HSP90AA1 P07900 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
MAPT P10636 2/20 0.39
S1PR1 P21453 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ATM Q13315 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
NOD2 Q9HC29 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035171 0.82 PYGL (0.45) PYGLNPC1RAB9AMEN1KMT2A
SCHEMBL8025608 0.81 CA12 (0.47) PYGLMAPTKDM4E
SCHEMBL8039185 0.80 PYGL (0.49) PYGLNPC1RAB9AMAPTMEN1
SCHEMBL8025601 0.80 TRPV1 (0.48) PYGLMAPT
SCHEMBL8037235 0.80 SMPD1 (0.45) PYGLNPC1RAB9AS1PR1KDM4E
SCHEMBL8041247 0.79 HSP90AA1 (0.39) HSP90AA1NPC1RAB9AMAPTMEN1
SCHEMBL8039096 0.79 PYGL (0.42) PYGLMEN1KMT2AKDM4E
SCHEMBL8039179 0.77 PYGL (0.46) PYGLNPC1RAB9AMAPTS1PR1
SCHEMBL8041323 0.77 KDM4E (0.45) PYGLMEN1KMT2AKDM4E
SCHEMBL8040249 0.75 PYGL (0.47) PYGLMAPTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed