SCHEMBL8041247

SCHEMBL8041247

COc1cc(Cl)c(C(=O)N(C)C(=O)NCC(F)(F)F)cc1O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.39
KMT2A Q03164 3/20 0.36
TRPV1 Q8NER1 1/20 0.35
CXCL12 P48061 2/20 0.34
BACE1 P56817 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GFER P55789 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
APP P05067 1/20 0.34
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
NOD2 Q9HC29 1/20 0.34
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8039016 0.85 HTT (0.42) HSP90AA1TRPV1CXCL12BACE1KDM4E
SCHEMBL8035589 0.83 TRPV1 (0.41) HSP90AA1KMT2ATRPV1CXCL12KDM4E
SCHEMBL8035119 0.81 KDM4E (0.40) HSP90AA1KMT2ACXCL12BACE1KDM4E
SCHEMBL8035099 0.81 TRPV1 (0.47) TRPV1
SCHEMBL8039231 0.80 CTSV (0.43) KMT2AKDM4EALDH1A1NPC1SMN1; SMN2
SCHEMBL8023948 0.79 PYGL (0.46) HSP90AA1KMT2AKDM4ENPC1MAPT
SCHEMBL8039002 0.78 MAPT (0.39) HSP90AA1KMT2ACXCL12KDM4EALDH1A1
SCHEMBL8039005 0.78 TRPV1 (0.41) HSP90AA1TRPV1ALDH1A1
SCHEMBL8025491 0.77 KDM4E (0.42) KMT2AKDM4EALDH1A1GFERL3MBTL1
SCHEMBL8032092 0.76 ALDH1A1 (0.44) KMT2AKDM4EALDH1A1GFERNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed