SCHEMBL8024749

SCHEMBL8024749

CC1(C)CSc2ccccc2NC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
PDK2 Q15119 1/20 0.44
PDK4 Q16654 1/20 0.44
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44
MEN1 O00255 6/20 0.43
KMT2A Q03164 6/20 0.43
GAA P10253 6/20 0.43
MAPT P10636 4/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALOX12 P18054 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
POLB P06746 2/20 0.42
CYP1A2 P05177 1/20 0.42
BCHE P06276 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ALOX15 P16050 1/20 0.42
MAOA P21397 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028203 0.80 ALDH1A1 (0.41) ALDH1A1PDK2PDK4BRD4CREBBP
SCHEMBL7745894 0.75 MEN1 (0.51) ALDH1A1PDK2PDK4BRD4CREBBP
SCHEMBL38579 0.73 ALDH1A1 (0.44) ALDH1A1BRD4CREBBPMEN1KMT2A
SCHEMBL29381975 0.73 ALDH1A1 (0.44) ALDH1A1BRD4CREBBPMEN1KMT2A
SCHEMBL8028186 0.73 KDM4E (0.36) ALDH1A1BRD4CREBBPMEN1KMT2A
SCHEMBL9629630 0.72 MEN1 (0.38) ALDH1A1PDK2PDK4BRD4CREBBP
SCHEMBL13323 0.71 ALDH1A1 (0.60) ALDH1A1PDK2BRD4CREBBPMEN1
SCHEMBL9148372 0.71 MAPT (0.37) ALDH1A1BRD4CREBBPMEN1KMT2A
SCHEMBL5999181 0.70 NPC1 (0.53) ALDH1A1PDK2PDK4BRD4CREBBP
Hydrochloric Acid SCHEMBL30648399 0.69 ALDH1A1 (0.58) ALDH1A1PDK2BRD4CREBBPMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed
EP-0792268-B1 HYPOLIPIDEMIC BENZOTHIAZEPINES WELLCOME FOUND (GB) 2000-02-23 EP disclosed
US-5998400-A Hypolipidemic benzothiazepines GLAXO WELLCOME INC. (US) 1999-12-07 US disclosed
EP-0792268-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1997-09-03 EP disclosed
WO-1996016051-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1996-05-30 WO disclosed