SCHEMBL8028203

SCHEMBL8028203

CCC1(CC)CSc2ccccc2NC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
POLB P06746 3/20 0.38
GAA P10253 6/20 0.37
MEN1 O00255 6/20 0.37
KMT2A Q03164 6/20 0.37
MAPT P10636 4/20 0.37
TDP1 Q9NUW8 3/20 0.37
CYP1A2 P05177 2/20 0.37
ALOX12 P18054 2/20 0.37
BCHE P06276 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ALOX15 P16050 1/20 0.37
MAOA P21397 1/20 0.37
CNR1 P21554 1/20 0.37
ACHE P22303 1/20 0.37
PTGS1 P23219 1/20 0.37
SLC6A2 P23975 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028186 0.89 KDM4E (0.36) ALDH1A1BRD4CREBBPPOLBGAA
SCHEMBL8024749 0.80 ALDH1A1 (0.46) ALDH1A1BRD4CREBBPPOLBGAA
SCHEMBL21585948 0.78 MAOB (0.57) ALDH1A1GAAMEN1KMT2AMAPT
SCHEMBL21586009 0.70 PTPN1 (0.37) ALDH1A1KMT2AHTR2CKDM4E
SCHEMBL8024372 0.69 MAOB (0.50) ALDH1A1GAAMEN1KMT2AMAPT
SCHEMBL22476283 0.69 KMT2A (0.43) POLBMEN1KMT2AMAPTHTR2C
SCHEMBL8024775 0.69 SLC6A2 (0.49) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL7745894 0.66 MEN1 (0.51) ALDH1A1BRD4CREBBPPOLBGAA
SCHEMBL13323 0.66 ALDH1A1 (0.60) ALDH1A1BRD4CREBBPPOLBGAA
SCHEMBL9817710 0.65 ALDH1A1 (0.47) ALDH1A1BRD4CREBBPPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792268-B1 HYPOLIPIDEMIC BENZOTHIAZEPINES WELLCOME FOUND (GB) 2000-02-23 EP disclosed
US-5998400-A Hypolipidemic benzothiazepines GLAXO WELLCOME INC. (US) 1999-12-07 US disclosed
EP-0792268-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1997-09-03 EP disclosed
WO-1996016051-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1996-05-30 WO disclosed