SCHEMBL8024781

SCHEMBL8024781

COc1ccc(CNc2ncnc(C(C)F)c2Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.55
CDK1 P06493 3/20 0.54
CCNB2 O95067 2/20 0.54
CCNB1 P14635 2/20 0.54
CCNB3 Q8WWL7 2/20 0.54
EGFR P00533 4/20 0.53
POLB P06746 2/20 0.53
NR2F2 P24468 1/20 0.53
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
PDE5A O76074 1/20 0.51
THRB P10828 2/20 0.49
MAPT P10636 3/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
KDM4E B2RXH2 2/20 0.46
MAPK1 P28482 2/20 0.46
OXTR P30559 1/20 0.46
BLM P54132 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037695 0.88 TP53 (0.51) HTTCDK1CCNB2CCNB1CCNB3
SCHEMBL8024318 0.87 EGFR (0.51) HTTEGFRPOLBPDE5AMAPT
SCHEMBL8025185 0.85 PRMT1 (0.48) HTTEGFRPOLBMEN1KMT2A
SCHEMBL8026802 0.84 CDK1 (0.50) HTTCDK1CCNB2CCNB1CCNB3
SCHEMBL29176418 0.79 HTT (0.43) HTTCDK1CCNB2CCNB1CCNB3
SCHEMBL8024930 0.78 EGFR (0.48) EGFRNR2F2AURKARPS6KB1
SCHEMBL9038905 0.78 TP53 (0.51) HTTCDK1CCNB2CCNB1CCNB3
SCHEMBL16997389 0.77 PDE5A (0.60) HTTEGFRPOLBMEN1KMT2A
Flufenerim SCHEMBL26581 0.75 CYP3A4 (0.42) HTTPOLBNR2F2MEN1KMT2A
Flufenerim SCHEMBL29429245 0.75 CYP3A4 (0.42) HTTPOLBNR2F2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543402-B1 Aralkylaminopyrimidine derivative, method for preparing the same and composition for controlling noxious organisms UBE INDUSTRIES (JP) 2000-03-01 EP claimed
US-5280025-A Aralkylaminopyrimidine derivative, and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1994-01-18 US claimed
EP-0543402-A1 Aralkylaminopyrimidine derivative, method for preparing the same and chemical for controlling noxious organisms containing the same UBE INDUSTRIES, LTD. (JP) 1993-05-26 EP claimed