SCHEMBL8024951

SCHEMBL8024951

O=C1CCC([C@H]2CC[C@H](c3ccc(-c4ccc(F)c(F)c4)cc3)CC2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.42
PGR P06401 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
P2RY14 Q15391 1/20 0.35
CYP17A1 P05093 2/20 0.35
CYP11B2 P19099 2/20 0.35
CYP3A4 P08684 1/20 0.35
NOTUM Q6P988 1/20 0.33
HSP90AA1 P07900 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM1A O60341 1/20 0.33
TNKS O95271 2/20 0.33
TNKS2 Q9H2K2 2/20 0.33
PTGS2 P35354 3/20 0.33
PTGS1 P23219 2/20 0.33
CYP11B1 P15538 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024950 1.00 ESR2 (0.42) ESR2PGRNPC1RAB9AP2RY14
SCHEMBL8379902 0.91 ESR2 (0.51) ESR2PGRNPC1RAB9AP2RY14
SCHEMBL7775189 0.88 ESR2 (0.43) ESR2KDM1APDE4APDE4BPDE4C
SCHEMBL7775191 0.88 ESR2 (0.43) ESR2KDM1APDE4APDE4BPDE4C
SCHEMBL8768421 0.84 PGR (0.39) PGRNPC1RAB9AP2RY14CYP17A1
SCHEMBL8768418 0.84 PGR (0.39) PGRNPC1RAB9AP2RY14CYP17A1
SCHEMBL19850903 0.83 KMT2A (0.39) PGRNPC1RAB9AP2RY14CYP17A1
SCHEMBL13345629 0.82 KDM1A (0.35) PGRNPC1RAB9AP2RY14CYP17A1
SCHEMBL14064159 0.82 ESR2 (0.46) ESR2PGRNPC1RAB9AP2RY14
SCHEMBL8015335 0.81 P2RY14 (0.33) PGRNPC1RAB9AP2RY14CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497176-B1 Four rings compounds and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 2000-04-05 EP disclosed
US-5478497-A For electro-optical purposes HOFFMANN-LA ROCHE INC. (US) 1995-12-26 US disclosed
EP-0497176-A2 Four rings compounds and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1992-08-05 EP disclosed