SCHEMBL8025554

SCHEMBL8025554

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NCCNC(C)=O)cc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HPGD P15428 1/20 0.41
APEX1 P27695 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
S1PR1 P21453 6/20 0.40
APP P05067 1/20 0.38
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
MAPK13 O15264 1/20 0.37
PDPK1 O15530 1/20 0.37
DAPK3 O43293 1/20 0.37
DYRK3 O43781 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037415 0.89 S1PR1 (0.41) MTNR1AHPGDS1PR1APPACHE
SCHEMBL8037435 0.87 PDE10A (0.41) S1PR1APP
SCHEMBL8037394 0.87 POLB (0.46) MTNR1AMTNR1BKDM4EHPGDS1PR1
SCHEMBL8037440 0.86 PDE10A (0.42)
SCHEMBL8035132 0.85 S1PR1 (0.38) KDM4ES1PR1APPACHE
SCHEMBL8037444 0.85 EPHX2 (0.43)
SCHEMBL8041448 0.85 EPHX2 (0.43)
SCHEMBL8041411 0.84 S1PR1 (0.43) KDM4ES1PR1APPACHE
SCHEMBL8035725 0.84 KDM4E (0.43) KDM4EHPGDS1PR1
SCHEMBL8041325 0.83 ALDH1A1 (0.45) KDM4ES1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed