SCHEMBL8041325

SCHEMBL8041325

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NCCCOC(C)C)cc1O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 3/20 0.45
POLB P06746 2/20 0.42
HTT P42858 2/20 0.42
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
S1PR1 P21453 1/20 0.39
TSHR P16473 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037394 0.91 POLB (0.46) ALDH1A1KDM4EPOLBS1PR1L3MBTL1
SCHEMBL8035725 0.87 KDM4E (0.43) ALDH1A1KDM4EPOLBHTTRAB9A
SCHEMBL8037435 0.86 PDE10A (0.41) S1PR1
SCHEMBL8037440 0.85 PDE10A (0.42)
SCHEMBL8037444 0.84 EPHX2 (0.43)
SCHEMBL8041448 0.84 EPHX2 (0.43)
SCHEMBL8037415 0.84 S1PR1 (0.41) ALDH1A1POLBS1PR1KMT2AMEN1
SCHEMBL8041411 0.83 S1PR1 (0.43) ALDH1A1KDM4EPOLBHTTS1PR1
SCHEMBL8025554 0.83 MTNR1A (0.42) KDM4ES1PR1
SCHEMBL8041695 0.82 MTNR1B (0.43) ALDH1A1KDM4EPOLBHTTS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed