SCHEMBL8037435

SCHEMBL8037435

CCCCNC(=O)NC(=O)c1cc(O)c(OC)cc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.41
FAAH O00519 1/20 0.40
S1PR1 P21453 3/20 0.39
NR5A2 O00482 1/20 0.38
NR5A1 Q13285 1/20 0.38
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037440 0.97 PDE10A (0.42) PDE10AFAAH
SCHEMBL8037444 0.96 EPHX2 (0.43) PDE10A
SCHEMBL8041448 0.96 EPHX2 (0.43) PDE10A
SCHEMBL8037415 0.93 S1PR1 (0.41) S1PR1APP
SCHEMBL8037394 0.91 POLB (0.46) S1PR1APP
SCHEMBL8035725 0.89 KDM4E (0.43) S1PR1
SCHEMBL8025554 0.87 MTNR1A (0.42) S1PR1APP
SCHEMBL8035132 0.87 S1PR1 (0.38) S1PR1APP
SCHEMBL8041325 0.86 ALDH1A1 (0.45) S1PR1
SCHEMBL8041411 0.83 S1PR1 (0.43) S1PR1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed