SCHEMBL8026248

SCHEMBL8026248

COc1ccc(B(O)O)cc1C1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HTR2C P28335 4/20 0.40
HTR2A P28223 4/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.37
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36
TUBB2B Q9BVA1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13687845 0.79 PTGDR2 (0.42) CA1CA2HTR2APTGDR2
SCHEMBL3790291 0.77 ENPP2 (0.40) ENPP2CA1CA2
SCHEMBL851880 0.76 ENPP2 (0.36) ENPP2CA1CA2TUBB4ATUBB
SCHEMBL23114 0.75 ENPP2 (0.52) ENPP2CA1CA2TUBB4ATUBB
SCHEMBL16957840 0.74 ACHE (0.54) HTR2CHTR2APTGDR2KMT2A
SCHEMBL16950302 0.74 HTR2C (0.41) CA1CA2HTR2CHTR2APTGDR2
SCHEMBL16957839 0.73 HTR2C (0.43) CA2HTR2CHTR2APTGDR2MEN1
SCHEMBL21231846 0.73 SLC6A2 (0.54) HTR2CHTR2APTGDR2
SCHEMBL3790241 0.73 ENPP2 (0.39) ENPP2CA1CA2
SCHEMBL7938441 0.73 KDM4E (0.46) HTR2CHTR2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089027-A1 PHOSPHODIESTERASE INHIBITORS GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICE, NATIONAL INSTITUTES OF HEALTH (US) 2009-07-16 WO disclosed