SCHEMBL8026513

SCHEMBL8026513

COC(=O)/C(=C/O)N(C)c1cccc(C(=N)OCc2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
RAB9A P51151 4/20 0.39
MAPT P10636 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PTPN1 P18031 1/20 0.35
NPC1 O15118 2/20 0.35
HTT P42858 1/20 0.35
MDM2 Q00987 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
SENP1 Q9P0U3 2/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009740 0.78 ALDH1A1 (0.42) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL8024358 0.78 L3MBTL1 (0.43) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL8024356 0.78 L3MBTL1 (0.43) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL27534529 0.77 ALDH1A1 (0.43) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL8026515 0.76 KMT2A (0.40) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL9456051 0.75 HSD17B2 (0.46)
SCHEMBL8020436 0.74 PPARG (0.48) RAB9ASMN1; SMN2HPGDKMT2AL3MBTL1
SCHEMBL8020434 0.72 PPARG (0.47) RAB9ASMN1; SMN2HPGDL3MBTL1NPC1
SCHEMBL29793626 0.69 MAOB (0.55) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD
SCHEMBL7770720 0.69 L3MBTL1 (0.44) ALDH1A1RAB9AMAPTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975587-A1 OXIME ETHER COMPOUNDS, THEIR USE AND INTERMEDIATES FOR PREPARATIONS OF THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2000-02-02 EP disclosed
WO-1998043949-A1 OXIME ETHER COMPOUNDS, THEIR USE AND INTERMEDIATES FOR PREPARATIONS OF THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-10-08 WO disclosed