SCHEMBL8026646

SCHEMBL8026646

O=C1COC(CC[N+]23CCC(c4ccccc4)(CC2)C3)(c2ccc(Cl)c(Cl)c2)CN1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.37
TACR2 P21452 2/20 0.36
TACR3 P29371 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630773 0.95 TACR1 (0.38) TACR1TACR2TACR3
Water SCHEMBL7749169 0.94 TACR1 (0.37) TACR1TACR2TACR3
SCHEMBL4631313 0.86 ADRB2 (0.37) TACR1TACR2
Water SCHEMBL7749198 0.85 ADRB2 (0.38) TACR1TACR2
SCHEMBL4631689 0.84 TACR1 (0.35) TACR1TACR2TACR3
Water SCHEMBL7744617 0.83 TACR1 (0.34) TACR1TACR2TACR3
SCHEMBL7764281 0.80 CCR5 (0.46) TACR1TACR2TACR3
SCHEMBL4631194 0.80 TACR1 (0.38) TACR1TACR2TACR3
SCHEMBL8456852 0.80 TACR1 (0.33) TACR1
SCHEMBL8991942 0.79 TACR1 (0.53) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011154-A Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present SANOFI (FR) 2000-01-04 US disclosed
EP-0915882-A1 1-AZONIABICYCLO[2.2.1]HEPTANE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (FR) 1999-05-19 EP disclosed
WO-1998004561-A1 1-AZONIABICYCLO[2.2.1]HEPTANE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (FR) 1998-02-05 WO disclosed