SCHEMBL8028096

SCHEMBL8028096

COc1cc(Cl)c(C(=O)N(C)C(=O)N(C(C)C)C(C)C)c([N+](=O)[O-])c1O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.35
POLB P06746 3/20 0.35
KDM4E B2RXH2 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
MAPT P10636 2/20 0.35
BLM P54132 2/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 1/20 0.34
ERN1 O75460 1/20 0.33
CDK2 P24941 1/20 0.33
TTR P02766 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
G6PD P11413 1/20 0.32
CRHBP P24387 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035686 0.86 COMT (0.38) TDP1POLBKDM4EL3MBTL1MAPT
SCHEMBL8041629 0.85 TDP1 (0.34) TDP1POLBKDM4EL3MBTL1CTDSP1
SCHEMBL8028100 0.83 L3MBTL1 (0.35) TDP1POLBKDM4EL3MBTL1CTDSP1
SCHEMBL8040095 0.82 ERN1 (0.37) TDP1POLBKDM4EL3MBTL1CTDSP1
SCHEMBL8044817 0.81 ALDH1A1 (0.35) TDP1POLBKDM4EL3MBTL1CTDSP1
SCHEMBL8041621 0.80 MEN1 (0.40) POLBKDM4EMAPTMEN1KMT2A
SCHEMBL8040090 0.79 GAA (0.42) KDM4EL3MBTL1MAPTMEN1KMT2A
SCHEMBL8038161 0.79 ERN1 (0.38) TDP1POLBKDM4EL3MBTL1CTDSP1
SCHEMBL8038657 0.78 POLB (0.40) POLBL3MBTL1MAPTMEN1KMT2A
SCHEMBL8041625 0.78 EGFR (0.35) TDP1POLBKDM4EL3MBTL1CTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed