SCHEMBL8028176

SCHEMBL8028176

C=C(c1ccc(C(=O)OC)cc1)c1ccc2c(c1)C(C)=C(C)CC2(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.43
RARG P13631 6/20 0.43
RXRA P19793 5/20 0.43
RARA P10276 4/20 0.43
RXRB P28702 2/20 0.43
RXRG P48443 2/20 0.43
CYP3A4 P08684 3/20 0.40
PDK2 Q15119 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
CYP26A1 O43174 3/20 0.38
POLB P06746 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026383 0.88 CYP3A4 (0.42) RARBRARGRXRARARARXRB
SCHEMBL8028154 0.86 RXRA (0.59) RARBRARGRXRARARARXRB
SCHEMBL6814364 0.82 PDK2 (0.40) RARBRARGRXRARARARXRB
SCHEMBL8028178 0.82 PTPN1 (0.50) RARBRARGRXRARARACYP3A4
SCHEMBL6814439 0.82 RARB (0.37) RARBRARGRXRARARARXRB
SCHEMBL8026629 0.81 RARB (0.43) RARBRARGRXRARARARXRB
SCHEMBL6814372 0.78 RXRA (0.49) RARBRARGRXRARARARXRB
SCHEMBL7421758 0.77 RXRA (0.72) RARBRARGRXRARARARXRB
SCHEMBL6814070 0.76 RARB (0.41) RARBRARGRXRARARARXRB
SCHEMBL8026052 0.75 RARB (0.41) RARBRARGRXRARARARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000059861-A1 SELECTIVE RETINOIC ACID ANALOGS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-10-12 WO disclosed