SCHEMBL8028665

SCHEMBL8028665

Fc1ccc2c(c1)CNCc1nccn1-2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 7/20 0.36
AVPR1A P37288 2/20 0.35
ROCK1 Q13464 2/20 0.35
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
ADRA2A P08913 1/20 0.32
ADRA1D P25100 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
EIF4E P06730 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
NOTUM Q6P988 1/20 0.31
NR3C2 P08235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029367 0.88 ADRA1A (0.36) ADRA1AAVPR1AROCK1HTR2CHTR2B
SCHEMBL8035211 0.82
SCHEMBL8032869 0.78 AVPR1A (0.41) ADRA1AAVPR1AADRA2A
SCHEMBL14996185 0.77 CYP11B2 (0.38) AVPR1AHTR2CHTR2BCYP1A2CYP2D6
SCHEMBL2062166 0.73 BTK (0.30)
SCHEMBL13002482 0.69 ROCK1 (0.35) ROCK1HTR2CHTR2BCYP1A2CYP2D6
SCHEMBL8030562 0.68 GABRG2 (0.39) CYP1A2CYP2D6NOTUM
SCHEMBL13002480 0.67 NOTUM (0.36) CYP1A2NOTUM
Hydrochloric Acid SCHEMBL2315581 0.66 CYP1A2 (0.41) HTR2CADRA2ACYP1A2CYP2D6
SCHEMBL107103 0.65 CYP1A2 (0.43) HTR2CADRA2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC PHARMA LIMITED (IN) 2010-12-09 US disclosed
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC PHARMA LIMITED (IN) 2010-12-09 US disclosed
WO-2009093269-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LIMITED (IN) 2009-07-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS DPP4, DPP3, DPP8 ADRA1A 1704/4885AVPR1A 369/4885ROCK1 3161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.