SCHEMBL8028680

SCHEMBL8028680

Nc1ccccc1NC(=O)/C=C/c1ccc(C(O)C(=O)O)cc1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.60
HDAC4 P56524 3/20 0.56
MEF2D Q14814 3/20 0.56
MMP1 P03956 2/20 0.53
MMP2 P08253 2/20 0.53
MMP9 P14780 2/20 0.53
EGFR P00533 1/20 0.53
HDAC2 Q92769 3/20 0.53
KDM1A O60341 1/20 0.52
MAOA P21397 1/20 0.52
EP300 Q09472 1/20 0.51
HDAC3 O15379 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978891 0.86 HDAC1 (0.60) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL3228591 0.85 EGFR (0.71) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL3228583 0.85 EGFR (0.71) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL2640602 0.82 HDAC1 (0.66) HDAC1MMP1MMP2MMP9EGFR
SCHEMBL7978520 0.81 HDAC1 (0.64) HDAC1MMP1MMP2MMP9EGFR
SCHEMBL4536420 0.80 TRPA1 (0.68) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL8348482 0.80 TRPA1 (0.68) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL13180844 0.80 HDAC1 (0.74) HDAC1HDAC4MMP1MMP2MMP9
SCHEMBL4536422 0.80 TRPA1 (0.68) HDAC1HDAC4MEF2DMMP1MMP2
SCHEMBL28633277 0.80 HDAC1 (0.63) HDAC1MMP1MMP2MMP9EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095324-A1 NOVEL N-(2-AMINO-PHENYL)-AMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-06 WO disclosed