SCHEMBL8028708

SCHEMBL8028708

CC(=O)C(=Cc1cc([N+](=O)[O-])c(O)c([N+](=O)[O-])c1)C(C)=O

nearest known ligand 0.85

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 3/20 0.85
GLO1 Q04760 1/20 0.54
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
RECQL P46063 1/20 0.49
KMT2A Q03164 1/20 0.49
XDH P47989 1/20 0.49
EGFR P00533 1/20 0.47
KDM4E B2RXH2 1/20 0.46
FTO Q9C0B1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitecapone SCHEMBL128420 0.92 GPR35 (1.00) GPR35GLO1ALDH1A1MEN1MAPT
Nitecapone SCHEMBL7039409 0.92 GPR35 (1.00) GPR35GLO1ALDH1A1MEN1MAPT
Nitecapone SCHEMBL30489171 0.92 GPR35 (1.00) GPR35GLO1ALDH1A1MEN1MAPT
SCHEMBL7279215 0.87 GPR35 (0.70) GPR35ALDH1A1MEN1MAPTKMT2A
SCHEMBL16884524 0.83 GPR35 (0.65) GPR35GLO1ALDH1A1MEN1MAPT
SCHEMBL9252649 0.81 GPR35 (0.62) GPR35GLO1ALDH1A1MEN1MAPT
SCHEMBL7287709 0.81 GPR35 (0.70) GPR35GLO1ALDH1A1MEN1MAPT
SCHEMBL7279195 0.79 GPR35 (0.78) GPR35ALDH1A1MEN1MAPTHPGD
SCHEMBL7279188 0.79 GPR35 (0.78) GPR35ALDH1A1MEN1MAPTHPGD
SCHEMBL8045644 0.79 GLO1 (0.71) GPR35GLO1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-5292771-A Treating inflammatory bowel disease ORION-YHTYMA OY (FI) 1994-03-08 US disclosed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP disclosed