SCHEMBL8045644

SCHEMBL8045644

CC(=O)C(=Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1)C(C)=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 3/20 0.71
GPR35 Q9HC97 1/20 0.59
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA4 P22748 1/20 0.45
CA7 P43166 1/20 0.45
ALDH1A1 P00352 4/20 0.44
CYP3A4 P08684 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP19A1 P11511 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
GLA P06280 1/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028846 0.83 GLO1 (1.00) GLO1GPR35CA1CA2CA4
SCHEMBL7245950 0.81 GLO1 (0.66) GLO1GPR35ALDH1A1SMN1; SMN2KDM4E
SCHEMBL8028708 0.79 GPR35 (0.85) GLO1GPR35ALDH1A1KDM4EMEN1
SCHEMBL9401844 0.76 GLO1 (0.86) GLO1CA1CA2CA4CA7
SCHEMBL7277503 0.76 GLO1 (0.86) GLO1CA1CA2CA4CA7
SCHEMBL7271725 0.76 GLO1 (0.86) GLO1CA1CA2CA4CA7
SCHEMBL7271722 0.76 GLO1 (0.86) GLO1CA1CA2CA4CA7
Nitecapone SCHEMBL7039409 0.75 GPR35 (1.00) GLO1GPR35ALDH1A1MEN1LMNA
Nitecapone SCHEMBL128420 0.75 GPR35 (1.00) GLO1GPR35ALDH1A1MEN1LMNA
Nitecapone SCHEMBL30489171 0.75 GPR35 (1.00) GLO1GPR35ALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP claimed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-5292771-A Treating inflammatory bowel disease ORION-YHTYMA OY (FI) 1994-03-08 US disclosed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP disclosed