SCHEMBL8028754

SCHEMBL8028754

O=C(O)c1ccc(C=C(C(=O)C2CC2)C(=O)C2CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
TDP1 Q9NUW8 2/20 0.58
POLB P06746 2/20 0.58
GLA P06280 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
RARG P13631 6/20 0.44
RARB P10826 5/20 0.44
MAPT P10636 5/20 0.43
HTT P42858 4/20 0.43
NPSR1 Q6W5P4 4/20 0.43
LMNA P02545 3/20 0.43
RAB9A P51151 3/20 0.43
ATM Q13315 2/20 0.43
NPC1 O15118 2/20 0.43
RECQL P46063 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
STAT1 P42224 1/20 0.43
KMT2A Q03164 3/20 0.43
TP53 P04637 2/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040507 0.76 RAB9A (0.49) ALDH1A1MAPTNPSR1RAB9AATM
SCHEMBL8040495 0.76 KMT2A (0.48) ALDH1A1L3MBTL1MAPTLMNARAB9A
SCHEMBL8876005 0.76 MEN1 (0.44) ALDH1A1POLBMAPTHTTNPSR1
SCHEMBL8876007 0.76 MEN1 (0.44) ALDH1A1POLBMAPTHTTNPSR1
SCHEMBL8038684 0.75 NAMPT (0.60) ALDH1A1TDP1L3MBTL1RARGMAPT
SCHEMBL2554589 0.73 ALDH1A1 (1.00) ALDH1A1TDP1POLBGLAL3MBTL1
SCHEMBL6885182 0.72 MAPT (0.54) ALDH1A1POLBGLAL3MBTL1MAPT
SCHEMBL7577513 0.72 ALDH1A1 (0.46) ALDH1A1TDP1POLBGLAL3MBTL1
Terephthalic Acid SCHEMBL6654100 0.72 TSHR (0.60) ALDH1A1MAPTLMNARAB9ANPC1
SCHEMBL2743573 0.70 SRD5A2 (0.71) ALDH1A1RAB9ANPC1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP claimed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP claimed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-5292771-A Treating inflammatory bowel disease ORION-YHTYMA OY (FI) 1994-03-08 US disclosed
US-5185370-A Substituted β-diketones and their use ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
EP-0440324-A2 Substituted beta-diketones and their use ORION-YHTYMÀ„ OY (FI) 1991-08-07 EP disclosed