SCHEMBL8031336

SCHEMBL8031336

COC(=O)c1ccc(C(=O)c2ccc3c(c2)C(C(C)C)=CCC3(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
RARB P10826 12/20 0.39
RARG P13631 10/20 0.39
RARA P10276 10/20 0.39
RXRA P19793 2/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
CYP26A1 O43174 2/20 0.37
PDK2 Q15119 1/20 0.37
NR2E1 Q9Y466 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026052 0.88 RARB (0.41) CYP3A4RARBRARGRARARXRA
SCHEMBL8026053 0.85 RARA (0.53) CYP3A4RARBRARGRARARXRA
SCHEMBL8026706 0.84 CYP3A4 (0.42) CYP3A4RARBRARGRARARXRA
SCHEMBL8028151 0.79 RARB (0.62) RARBRARGRARARXRANR2E1
SCHEMBL8032216 0.75 RARB (0.55) RARBRARGRARARXRARXRB
SCHEMBL8026383 0.74 CYP3A4 (0.42) CYP3A4RARBRARGRARARXRA
SCHEMBL6086597 0.73 RARB (0.44) RARBRARGRARAMAPTPDK2
SCHEMBL7422927 0.72 RXRA (0.70) CYP3A4RARBRARGRARARXRA
SCHEMBL8026629 0.72 RARB (0.43) CYP3A4RARBRARGRARARXRA
SCHEMBL6810972 0.72 RARA (0.39) CYP3A4RARBRARGRARARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000059861-A1 SELECTIVE RETINOIC ACID ANALOGS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-10-12 WO disclosed